1. シグナル伝達
  2. Epigenetics
  3. Histone Acetyltransferase
  4. Histone Acetyltransferase Inhibitors

Histone Acetyltransferase Inhibitors

CBP/p300

GCN5/PCAF

TIP60

MOZ/MORF

HBO1

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Histone Acetyltransferase Inhibitors, Activators, Degraders & Ligands
製品名 CBP/p300 GCN5/PCAF TIP60 MOZ/MORF HBO1 純度
A-485
CBP/p300
        99.87%
Curcumin
CBP/p300
        98.84%
C646
CBP/p300
        99.88%
WM-3835        
HBO1
99.78%
JZY3032
p300
       
SGC-CBP30
CBP/p300
        99.83%
PF-9363      
MOZ/MORF
  99.64%
MG 149
CBP/p300
 
TIP60
    99.60%
Butyrolactone 3  
GCN5, IC50: 100 μM
      99.58%
Anacardic Acid
p300-HAT, IC50: 8.5 μM
PCAF, IC50: 5 μM
      98.49%
CTB
CBP/p300
        99.93%
WM-8014      
MOZ/MORF
  99.92%
WM-1119      
MOZ/MORF
  99.57%
NSC 228155
KIX-KID, IC50: 0.36 μM
       
Garcinol  
GCN5/PCAF
      98.85%
GNE-049
CBP/p300
        99.74%
Prifetrastat  
GCN5/PCAF
      99.63%
CPI-1612
CBP/p300
        99.75%
PU139
CREBBP, IC50: 2.49 μM
p300, IC50: 5.35 μM
GCN5, IC50: 8.39 μM
PCAF, IC50: 9.74 μM
      99.51%
TTK21
CBP/p300
        99.39%
CPTH2  
GCN5
      99.82%
GSK 4027  
GCN5/PCAF
      98.22%
CTPB
CBP/p300
        ≥99.0%
NEO2734
CBP/p300
        99.63%
GNE-272
CBP/p300
        99.60%
TH1834    
TIP60
    99.79%
AUR1545  
GCN5/PCAF
      99.58%
I-CBP112
CBP/p300
        98.43%
GNE-207
CBP, IC50: 1 nM
        99.94%
YF-2
CBP, EC50: 2.75 μM
GCN5, EC50: 49.31 μM
GCN5/PCAF, EC50: 29.04 μM
      98.76%
Procyanidin B3
CBP/p300
        99.92%
TH1834 dihydrochloride    
TIP60
    99.89%
JET-209
CBP, DC50: 0.05 nM
p300, DC50: 0.2 nM
        98.07%
L002
CBP/p300
        99.44%
Histone Acetyltransferase Inhibitor II
CBP/p300
        98.70%
GSK699  
GCN5/PCAF
      98.80%
GSK4028  
GCN5/PCAF
      98.06%
Curcumin-d6
CBP/p300
        99.78%
PCAF-IN-2  
PCAF, IC50: 5.31 μM
      98.0%
CBP/p300-IN-3
CBP/p300
        98.01%
Lys-CoA TFA
p300, IC50: 50-500 nM
        98.52%
YF-2 hydrochloride
CBP, EC50: 2.75 μM
GCN5, EC50: 49.31 μM
GCN5/PCAF, EC50: 29.04 μM
      99.29%
TPOP146
CBP/p300
        98.94%
DCH36_06
CBP/p300
        99.19%
NSC 694623  
PCAF, IC50: 15.9 μM
      99.53%
CBP/p300-IN-12
CBP/p300, IC50: 166 nM
        99.72%
Naphthol AS-E
KIX-KID, IC50: 2.26 μM
        98.0%
MOZ-IN-2      
MOZ/MORF
  99.58%
CBP/p300-IN-19 hydrochloride
p300-HAT, IC50: 1.4 μM
CBP-HAT, IC50: 2.2 μM
PCAF, IC50: >100 μM
      99.00%
KAT6A/KAT7-IN-4      
MOZ/MORF, IC50: <1 nM
HBO1, IC50: <1 nM
98.86%
CBP/p300-IN-10
EP300, IC50: 26 nM
CREBBP, IC50: 39 nM
        99.74%
NiCur
CBP-HAT, IC50: 0.35 μM
        99.11%
BT-O2C
p300
       
CBP/p300-IN-5
CBP/p300
       
B026
p300, IC50: 8.1 nM
CBP, IC50: 9.5 nM
       
CBP/p300-IN-20
CBP/p300, pIC50: 10.1
        98.03%
CAY10669  
PCAF, IC50: 662 μM
      99.9%
CPTH2 hydrochloride  
GCN5
     
DS17701585
EP300, IC50: 0.04 μM
CBP, IC50: 0.15 μM
       
CBP/p300-IN-14
CBP/p300
       
CBP/p300-IN-18
EP300, IC50: .056 μM
       
Ep300/CREBBP-IN-4
EP300, IC50: 0.024 μM
CREBBP, IC50: 0.064 μM
       
PROTAC KAT6 Degrader-1      
MOZ/MORF
 
CBP/p300-IN-15
CBP, IC50: 28 nM
p300, IC50: 2.5 nM
       
Ep300/CREBBP-IN-3
EP300, IC50: 0.056 μM
CREBBP, IC50: 0.095 μM
       
P300 bromodomain-IN-1
p300, IC50: 49 nM
       
PROTAC CBP/p300/BRD4 Degrader-1
CBP, DC50: 6.55 nM
p300, DC50: 1.05 nM
CBP, IC50: 110.8 nM
p300, IC50: 102.6 nM
       
PROTAC CBP/P300 Degrader-4
CBP, DC50: 10.2 nM
p300, DC50: 17.4 nM
       
CBP/p300/BRD4 ligand-1
CBP
p300
       
ACTR-AD1 2L
CBP/p300
       
Ep300/CREBBP-IN-2
EP300, IC50: 0.052 μM
CREBBP, IC50: 0.148 μM
       
CBP/p300-IN-17
EP300, IC50: .18 μM
       
GSK702  
PCAF
     
SL010110
p300
       
P300-IN-6
p300-HAT, IC50: 7 nM
       
ZX079
CBP
p300
       
PRMT/HKMT-IN-1
CBP/p300
       
Ep300/CREBBP-IN-8
EP300, IC50: 0.014 μM
CREBBP, IC50: 0.018 μM
       
CCT077791
p300
PCAF
     
CBP/p300-IN-22
CBP/p300, IC50: 4 nM
       
CBP/p300-IN-19
p300-HAT, IC50: 1.4 μM
CBP-HAT, IC50: 2.2 μM
PCAF, IC50: >100 μM
     
PROTAC MLT Degrader 1
p300
       
KAT2A/B ligand 1  
GCN5/PCAF
     
KCN1
p300